Course Information


Course Information
Course Title Code Semester L+U Hour Credits ECTS
DRUG DESIGN METHODS 34103009 2 + 0 2.0 6.0

Prerequisites None

Language of Instruction Turkish
Course Level Graduate Degree
Course Type Compulsory
Mode of delivery theoretical
Course Coordinator
Instructors
Assistants
Goals Gains information about designing methods of drug active compounds.
Course Content Studies on investigation and development of active compounds, relationships of effector and target, QSAR, physicochemical parameterization, Hansch analysis methods, Bilinear analysis methods, Free-Wilson modified analysis methods, Relationships between FujitaBan and Hansch models, Applications about models
Learning Outcomes 1) In development studies of drug active compounds, gains basic information about medicinal chemistry and drug design methods.
2) Practise drug design, synthesis, structure elucidation and analyses studies.
3) Gains information about designing methods of drug active compounds.

Weekly Topics (Content)
Week Topics Teaching and Learning Methods and Techniques Study Materials
1. Week Research and development studies for drug active compounds Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
2. Week Effector-target relationship Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
3. Week Effector-target relationship Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
4. Week QSAR Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
5. Week Physicochemical parametrization Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
6. Week Physicochemical parametrization Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
7. Week Midterms Question Answer

 Presentation (Including Preparation Time)
8. Week Hansch Analyses Method Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
9. Week Bilineer Analyses Method Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
10. Week Free-Wilson Analyses Method Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
11. Week Relationships between FujitaBan and Hansch Model Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
12. Week Practises of models Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
13. Week Practises of models Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
14. Week Practises of models Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
15. Week Practises of models Lecture; Question Answer; Discussion

 Activity (Web Search, Library Work, Trip, Observation, Interview etc.)
16. Week Final exam Question Answer

 Presentation (Including Preparation Time)

Sources Used in This Course
Recommended Sources
3D Qsar in Drug Design: Recent Advances, Gerd Folkers, 1998 Kluwer Academic Publishers
3D Qsar in Drug Design: Theory Methods and Applications, Hugo Kubinyi, 1993 Kluwer Academic Publishers
Evolutiory Algorithms in Molecular Design, Clark, D.E. (ED), Wiley-VCH, Weinheim, 2000.

Relations with Education Attainment Program Course Competencies
Program RequirementsContribution LevelDK1DK2DK3
PY15000
PY25000
PY35000
PY45000

*DK = Course's Contrubution.
0 1 2 3 4 5
Level of contribution None Very Low Low Fair High Very High
.

ECTS credits and course workload
Event Quantity Duration (Hour) Total Workload (Hour)
Course Duration (Total weeks*Hours per week) 1 1
Homework 5 5
Presentation (Including Preparation Time) 10 10
Report (Including Preparation and presentation Time) 5 5
Time to prepare for Quiz 5 5
Total Workload
Total Workload / 30 (s)
ECTS Credit of the Course
Quick Access Hızlı Erişim Genişlet
Course Information
  • Course Information
  • Weekly Topics (Content)
  • Sources Used in This Course
  • Relations with Education Attainment Program Course Competencies
  • ECTS credits and course workload